VU6043653

VU6043653 is a potent, selective and cross the blood-brain barrier metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 value of 325 nM for h mGlu5.


Cat. No.: EX-A12129	Purity: >98%

	Chemical structure of VU6043653

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	305	In-stock
250mg	610	In-stock
500mg	960	In-stock
1g	1560	In-stock
2g	2480	In-stock
3g	2980	In-stock

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CAS No.	3032791-06-0
Purity	>98%
Formula	C16H14FN5O2
Mol Weight	327.3131
Color	Off-white to light yellow
State	Solid
Solubility	DMSO : ? 25 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder 4°C, protect from light, stored under nitrogen; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Elizabeth S. Childress, et al. Discovery of 4-(5-Membered)Heteroarylether-6-methylpicolinamide Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5. ACS Med. Chem. Lett. 2024.
CoA	CoA of VU6043653

Smiles:	O=C(NC1=NC=C(F)C=C1)C=2N=C(C=C(OC=3C=NN(C3)C)C2)C


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