UK-78,282 hydrochloride

UK-78282, a novel piperidine, potent and selective Kv1.3 blocker with an IC50 of 200 nM. UK-78,282 effectively suppresses human T-lymphocyte activation in vitro. UK-78,282 binds to residues at the inner surface of the channel overlapping the site of action of verapamil[1].


Cat. No.: EX-A15260	Purity: >98%

	Chemical structure of UK-78,282 hydrochloride

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	459	in_stock
500mg	735	in_stock
1g	1181	in_stock
2g	1886	in_stock
3g	2299	in_stock
5g	2967	in_stock

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CAS No.	136647-02-4
Purity	>98%
Formula	C29H36ClNO2
Mol Weight	466.055
Color	White to off-white
State	Solid
Solubility	soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20°C, sealed storage, away from moisture; In solvent -20℃, 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. D C Hanson, et al. UK-78,282, a novel piperidine compound that potently blocks the Kv1.3 voltage-gated potassium channel and inhibits human T cell activation. Br J Pharmacol. 1999 Apr;126(8):1707-16
CoA	CoA of UK-78,282 hydrochloride

Smiles:	COC1=CC=C(C=C1)CCCN2CCC(CC2)COC(C3=CC=CC=C3)C4=CC=CC=C4.Cl


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