Tilfrinib

Tilfrinib (compound 4f) is a potent and selective Brk/PTK6 inhibitor with an IC50 value of 3.15 nM for Brk. Tilfrinib shows good anti-proliferative activity and has potential of anti-tumour .


Cat. No.: EX-A10268	Purity: >98%

	Chemical structure of Tilfrinib

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	700	In-stock
500mg	1300	In-stock
1g	2300	In-stock

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CAS No.	1600515-49-8
Purity	>98%
Formula	C17H13N3O
Mol Weight	275.3046
Color	off-white to yellow
State	solid
Solubility	Soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder 4℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Zhang Q, Liu S, et al. ETV4 mediated tumor-associated neutrophil recruitment promotes lymphangiogenesis and lymphatic metastasis of bladder cancer[J]. 2022. [2]. Mahmoud KA, et al. Discovery of 4-anilino α-carbolines as novel Brk inhibitors. Bioorg Med Chem Lett. 2014 Apr 15;24(8):1948-51.
CoA	CoA of Tilfrinib

Smiles:	OC1=CC=CC(NC2=C3C4=CC=CC=C4NC3=NC=C2)=C1


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