TAK-041

TAK-041 (Zelatriazin; NBI-1065846) is a potent and selective GPR139 agonist with an EC50 of 22 nM. TAK-041 has the potential for the research of negative symptoms associated with schizophrenia .


Cat. No.: EX-A6066	Purity: >98%

	Chemical structure of TAK-041

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
1g	932	in_stock
2g	1432	in_stock
5g	3264	inquire

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Synonyms	Zelatriazin
Synonyms 2	NBI-1065846
CAS No.	1929519-13-0
Purity	>98%
Formula	C18H15F3N4O3
Mol Weight	392.3319
Color	White to off-white
State	solid powder
Solubility	Soluble in DMSO 100 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder 4℃ 2 years; -20℃ 3 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Reichard, Holly A et al. “Discovery of TAK-041: a Potent and Selective GPR139 Agonist Explored for the Treatment of Negative Symptoms Associated with Schizophrenia. Journal of medicinal chemistry vol. 64,15 (2021): 11527-11542.
CoA	CoA of TAK-041

Smiles:	O=C(N[C@H](C1=CC=C(OC(F)(F)F)C=C1)C)CN2N=NC3=CC=CC=C3C2=O


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