T-10418

T-10418 is a potent and highly selective G2A/GPR132 agonist. T-10418 has an EC50 of 0.82 μM for human G2A activation. T-10418 has good water solubility, metabolic stability, and pharmacokinetic properties. T-10418 can be used for the research of various diseases such as neuropathic pain, acute myeloid leukemia, and inflammation .


Cat. No.: EX-A9944	Purity: >98%

	Chemical structure of T-10418

For research only, Do not use for Human!

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CAS No.	1608784-68-4
Purity	>98%
Formula	C22H20N2O4
Mol Weight	376.4052
Color	White to off-white
State	Solid
Solubility	Soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20℃ 3 years, 4℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Hernandez-Olmos V, et al., Development of a Potent and Selective G2A (GPR132) Agonist. J Med Chem. 2024 Jun 25.
CoA	CoA of T-10418

Smiles:	C(N[C@H](CC1=CC=CC=C1)C(O)=O)(=O)C2=CC(OCC=3C=CC=NC3)=CC=C2


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