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Product Information:

SR144528

SR144528 is a potent and selective CB2 receptor antagonist with a Ki of 0.6 nM.

Cat. No.: EX-A7261    Purity: >98%
Chemical
Chemical structure of SR144528


For research only, Do not use for Human!

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SynonymsSR 144528
CAS No.192703-06-3
Purity>98%
FormulaC29H34ClN3O
Mol Weight476.053
ColorWhite to light yellow
Statesolid powder
SolubilityDMSO : 100 mg/mL
Shelf Life>3 years if stored properly
StoragePowder -20°C, 3 years , 4°C, 2 years ; In solvent -20°C, 1 year
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1].Rinaldi-Carmona M, et al. SR 144528, the first potent and selective antagonist of the CB2 cannabinoid receptor. J Pharmacol Exp Ther. 1998 Feb;284(2):644-50.

[2].Thewke D, et al. AM-251 and SR144528 are acyl CoA:cholesterol acyltransferase inhibitors. Biochem Biophys Res Commun. 2009 Apr 3;381(2):181-6.

[3].Abalo R, et al. The cannabinoid antagonist SR144528 enhances the acute effect of WIN 55,212-2 on gastrointestinal motility in the rat. Neurogastroenterol Motil. 2010 Jun;22(6):694-e206.

CoACoA of SR144528

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