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Product Information:

BQ-123

BQ-123 is a selective endothelin A receptor (ETA) antagonist with IC50 of 7.3 nM.

Cat. No.: EX-A4062    Purity: >98%
BQ-123
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
50mg785In-stock
100mg1185In-stock
200mg1785In-stock
1gget quoteIn-stock


CAS No.136553-81-6
Purity>98%
FormulaC31H42N6O7
Mol Weight610.7012
Appearancesolid powder
SolubilitySoluble in DMSO
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Ihara, M et al. “In vitro biological profile of a highly potent novel endothelin (ET) antagonist BQ-123 selective for the ETA receptor. Journal of cardiovascular pharmacology vol. 20 Suppl 12 (1992): S11-4.

[2]. Eguchi, S et al. “A novel ETA antagonist (BQ-123) inhibits endothelin-1-induced phosphoinositide breakdown and DNA synthesis in rat vascular smooth muscle cells. FEBS letters vol. 302,3 (1992): 243-6.

CoACoA of BQ-123
Smiles:O=C(N[C@](C(N(CCC1)[C@]1([H])C2=O)=O)([H])CC(O)=O)[C@H](NC([C@@H](NC([C@H](N2)C(C)C)=O)CC(C)C)=O)CC3=CNC4=CC=CC=C34

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