VU6012962

VU6012962 is an orally bioavailable and CNS-penetrant metabotropic glutamate receptor 7 negative allosteric modulator (mGlu7 NAM) with an IC50 of 347 nM.


Cat. No.: EX-A2982	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
500mg	850	In-stock
1g	1300	In-stock
5g	4050	inquire

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CAS No.	2313526-86-0
Purity	>98%
Formula	C21H19F3N4O4
Mol Weight	448.3952
Appearance	off-white solid powder
Solubility	DMSO >100 mg/mL; Insoluble in water
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Reed CW, et al. Discovery of an orally bioavailable and Central Nervous System (CNS) penetrant mGlu7 NegativeAllosteric Modulator (NAM) in vivo tool compound: N-(2-(1H-1,2,4-triazol-1-yl)-5-(trifluoromethoxy)phenyl)-4-(cyclopropylmethoxy)-3-methoxybenzamide (VU6012962). J Med Chem. 2019 Jan 4.
CoA	CoA of VU6012962

Smiles:	COC1=CC(=CC=C1OCC1CC1)C(=O)NC1=C(C=CC(OC(F)(F)F)=C1)N1C=NC=N1


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