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Product Information:

GSK-2807 Trifluoroacetate

GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.

Cat. No.: EX-A3027    Purity: >98%
GSK-2807
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg985inquire
200mg1585In-stock
500mg2585In-stock
1g3885In-stock


SynonymsGSK2807 Trifluoroacetate
CAS No.2245255-66-5
Purity>98%
FormulaC21H33F3N8O7
Mol Weight566.5313
AppearancePowder
SolubilitySoluble in DMSO, not in water
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Van Aller GS, et al. Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets. Structure. 2016 May 3;24(5):774-781.

[2]. Kaniskan HÜ, et al. Inhibitors of Protein Methyltransferases and Demethylases. Chem Rev. 2018 Feb 14;118(3):989-1068.

CoACoA of GSK-2807 Trifluoroacetate
Smiles:OC(=O)C(F)(F)F.CN(C)CCCN(CC[C@H](N)C(O)=O)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)N1C=NC2=C(N)N=CN=C12

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