LSZ-102

LSZ-102 is a potent, orally bioactive and selective ERα antagonist and SERD (estrogen receptor degrader) with an IC50 of 0.2 nM has the potential for the treatment of Estrogen Receptor Positive Breast Cancer.


Cat. No.: EX-A1874	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	900	In-stock
100mg	1300	In-stock
200mg	1950	In-stock
1g	5200	In-stock
2g	8200	In-stock
5g	13500	Inquire

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Synonyms	LSZ102
Synonyms 2	SERD LSZ102
CAS No.	2135600-76-7
Purity	>98%
Formula	C25H17F3O4S
Mol Weight	470.46
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Tria GS, et al. Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer. J Med Chem. 2018 Apr 12;61(7):2837-2864.
CoA	CoA of LSZ-102

Smiles:	CC(F)(F)C1=CC(F)=CC=C1C1=C(OC2=CC=C(\C=C\C(O)=O)C=C2)C2=CC=C(O)C=C2S1


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