background


Product Information:

PF-4136309

PF-4136309 is a potent, selective, and orally bioavailable CCR2 antagonist, with IC50s of 5.2 nM, 17 nM and 13 nM for human, mouse and rat CCR2.

Cat. No.: EX-A2696    Purity: >98%
PF-4136309
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg500In-stock
250mg785In-stock
500mg1085In-stock
1g1685In-stock
2g2500In-stock
5g6685In-stock


SynonymsINCB8761
Synonyms 2857679-55-1
CAS No.1341224-83-6
Purity>98%
FormulaC29H31F3N6O3
Mol Weight568.59
Appearancesolid powder
SolubilitySoluble in DMSO/Ethanol
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Xue CB, et al. Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist. ACS Med. Chem. Lett., 2011, 2 (12), pp 913-918.

CoACoA of PF-4136309
Smiles:[H][C@@]1(CC[C@](O)(CC1)C1=NC=C(C=C1)C1=NC=CC=N1)N[C@H]1CCN(C1)C(=O)CNC(=O)C1=CC=CC(=C1)C(F)(F)F

KEYWORDS: buy PF-4136309 | PF-4136309 supplier | purchase | cost | manufacturer | order | distributor | buy 1341224-83-6 | 1341224-83-6 supplier