TG4-155

TG4-155 is a potent, brain-permeant and selective EP2 receptor antagonist with a Ki of 9.9 nM. TG4-155 shows low nanomolar antagonist activity against only EP2 and DP1[1]. TG4-155 has an EP2 Schild KB of 2.4 nM and displays 550-4750-fold selectivity for EP2 over EP1, EP3, EP4 and IP, but only 14-fold selectivity against the DP1 receptor.


Cat. No.: EX-A2930	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	585	In-stock
200mg	985	In-stock
1g	1885	In-stock
2g	3300	In-stock
5g	4650	In-stock

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CAS No.	1164462-05-8
Purity	>98%
Formula	C23H26N2O4
Mol Weight	394.4635
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Jiang J, et al. Role of prostaglandin receptor EP2 in the regulations of cancer cell proliferation, invasion, and inflammation. J Pharmacol Exp Ther. 2013 Feb;344(2):360-7. [2]. Ganesh T. Prostanoid receptor EP2 as a therapeutic target. J Med Chem. 2014 Jun 12;57(11):4454-65.
CoA	CoA of TG4-155

Smiles:	COC1=CC(\C=C\C(=O)NCCN2C(C)=CC3=CC=CC=C23)=CC(OC)=C1OC


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