Mirogabalin besylate

Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.


Cat. No.: EX-A2817	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	385	In-stock
250mg	485	In-stock
500mg	600	In-stock
1g	800	In-stock
2g	1200	In-stock
5g	2000	In-stock

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Synonyms	DS 5565 besylate
CAS No.	1138245-21-2
Purity	>98%
Formula	C18H25NO5S
Mol Weight	367.46
Appearance	White to off-white solid
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Domon Y, et al. Binding Characteristics and Analgesic Effects of Mirogabalin, a Novel Ligand for the α2δ Subunit of Voltage-Gated Calcium Channels. J Pharmacol Exp Ther. 2018 Jun;365(3):573-582.
CoA	CoA of Mirogabalin besylate

Smiles:	OS(=O)(=O)C1=CC=CC=C1.[H][C@@]12C[C@](CN)(CC(O)=O)[C@]1([H])C=C(CC)C2


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