RGH-122

RGH-122 (compound 43) is an orally active, potent, selective, and hV1a receptor antagonist with Ki value of 0.3 nM and IC50 of 0.9 nM. RGH-122 showes microsomal stability with CLint value of 13/28/25 μL/min/mg.


Cat. No.: EX-A14109	Purity: >98%

	Chemical structure of RGH-122

For research only, Do not use for Human!

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CAS No.	2355304-05-9
Purity	>98%
Formula	C24H25ClN4O3
Mol Weight	452.933
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Baska F, et al. Discovery and Characterization of RGH-122, a Potent, Selective, and Orally Bioavailable V1a Receptor Antagonist. J Med Chem. 2024 Jan 11;67(1):643-673.
CoA	CoA of RGH-122

Smiles:	ClC1=CC=[C@]2[N@]3C([C@H](CC4)CC[C@@H]4OC5=NC=CC=C5)=NN=C3CC6(OCCO6)CC2=C1


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