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Product Information:

Revefenacin

Revefenacin (TD-4208; GSK1160724) is a potent mAChR antagonist; has a high affinity on M3 receptor with a Ki of 0.18 nM.

Cat. No.: EX-A1722    Purity: >98%
Chemical
Chemical structure of Revefenacin


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
50mg360in_stock
100mg578in_stock
250mg1136in_stock
500mg1795in_stock
1g2972in_stock
2g4753in_stock


SynonymsTD-4208
Synonyms 2GSK1160724
CAS No.864750-70-9
Purity>98%
FormulaC35H43N5O4
Mol Weight597.747
Colorwhite to off-white
Statesolid powder
SolubilitySoluble in DMSO
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Steinfeld T, et al. In vitro characterization of TD-4208, a lung-selective and long-acting muscarinic antagonist bronchodilator (Abstract). Am J Respir Crit Care Med 179:A4553.

[2]. Pulido-Rios MT, et al. In vivo pharmacological characterization of TD-4208, a novel lung-selective inhaled muscarinic antagonist with sustained bronchoprotective effect in experimental animal models. J Pharmacol Exp Ther. 2013 Aug;346(2):241-50.

CoACoA of Revefenacin
Smiles:CN(CCN1CCC(CC1)OC(=O)NC1=CC=CC=C1C1=CC=CC=C1)C(=O)C1=CC=C(CN2CCC(CC2)C(N)=O)C=C1

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