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Product Information:

(Rac)-INCB8761

(Rac)-PF-4136309 is an isoform of PF-4136309 (EX-A2696), which is a potent, selective, and orally bioavailable CCR2 antagonist, with IC50s of 5.2 nM, 17 nM and 13 nM for human, mouse and rat CCR2.

Cat. No.: EX-A6109    Purity: >98%
Chemical
Chemical structure of (Rac)-INCB8761


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
500mg1050In-stock
1g1650In-stock
5g5600Inquire


Synonyms(Rac)-PF-4136309
Synonyms 21341224-83-6
CAS No.857679-55-1
Purity>98%
FormulaC29H31F3N6O3
Mol Weight568.59
ColorLight yellow to yellow
Statesolid powder
SolubilitySoluble in DMSO/Ethanol
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Xue CB, et al. Discovery of INCB8761/PF-4136309, a Potent, Selective, and Orally Bioavailable CCR2 Antagonist. ACS Med. Chem. Lett., 2011, 2 (12), pp 913-918.

CoACoA of (Rac)-INCB8761

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