PSMA-Val-Cit-PAB-Azide

PSMA-azide is a prostate-specific membrane antigen (PSMA) ligand. PSMA-azide inhibits PSMA-dependent NAAG (N-acetylaspartylglutamic acid) hydrolysis, with an IC50 of 9 nM and a Ki of 1 nM. PSMA-azide contains an Azide group and can undergo copper-catalyzed azide-alkyne cycloaddition reaction (CuAAc) with molecules containing Alkyne groups.


Cat. No.: EX-A17052	Purity: >98%

	Chemical structure of PSMA-Val-Cit-PAB-Azide

For research only, Do not use for Human!

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Synonyms	PSMA-azide
CAS No.	2374814-84-1
Purity	>98%
Formula	C50H65ClN10O13
Mol Weight	1049.563
Color	White to off-white
State	Solid
Solubility	DMSO : 200 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder -20°C 3 years, 4°C 2 years; In solvent -20°C, 1 month.
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Machulkin AE, et al. Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them. J Med Chem. 2021 Apr 22;64(8):4532-4552.
CoA	CoA of PSMA-Val-Cit-PAB-Azide

Smiles:	O=C(N[C@H](C(NCCCN=[N+]=[N-])=O)CC(C=C1)=CC=C1O)[C@@H](NC(CCC(NCCCCCC(N(CCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O)CC2=CC(Cl)=CC=C2)=O)=O)=O)CC3=CC=CC=C3


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