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Product Information:

PROTAC BET-bindingmoiety 1

PROTAC BET-binding moiety 1 is a key intermediate for the synthesis of high-affinity BET inhibitors .

Cat. No.: EX-A16475    Purity: >98%
Chemical
Chemical structure of PROTAC BET-bindingmoiety 1


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
25mg995In-stock
50mg1685In-stock
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SynonymsPROTAC BET-binding moiety 1
CAS No.2093387-77-8
Purity>98%
FormulaC25H25N7O4
Mol Weight487.5105
Colorlight yellow to yellow
Statesolid
Solubilitysoluble in DMSO
Shelf Life>3 years if stored properly
StoragePowder 4℃, 2 years; -20℃, 3 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Zhou B, et al. Discovery of a Small-Molecule Degrader of Bromodomain and Extra-Terminal (BET) Proteins with Picomolar Cellular Potencies and Capable of Achieving Tumor Regression. J Med Chem. 2018 Jan 25;61(2):462-481.

CoACoA of PROTAC BET-bindingmoiety 1
Smiles:CCN1C(=CC(=N1)C2CC2)NC3=NC(=NC4=C3C5=CC(=C(C=C5N4)C6=C(ON=C6C)C)OC)C(=O)O

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