Piperacetazine

Piperacetazine is an orally active dopamine receptor antagonist and phenothiazine antipsychotic. Piperacetazine can directly bind to the PAX3::FOXO1 fusion protein and inhibit its transcriptional activity. Piperacetazine also exhibits antitumor activity with an IC50 of 7.627 μM against PANC-1 cells. Piperacetazine can be used for the research of diseases such as schizophrenia and pancreatic cancer and other tumors.


Cat. No.: EX-A12259	Purity: >98%

	Chemical structure of Piperacetazine

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock	Quantity	Order
1g	980	In-stock
5g	2680	10

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Synonyms	SC 9794
CAS No.	3819-00-9
Purity	>98%
Formula	C24H30N2O2S
Mol Weight	410.572
Color	Light yellow to yellow
State	Solid
Solubility	Ethanol : 50 mg/mL DMSO : ? 6 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder -20°C, 3 years , 4°C, 2 years; In solvent -20℃ 1 year;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Nakazawa K, et al. Piperacetazine Directly Binds to the PAX3::FOXO1 Fusion Protein and Inhibits Its Transcriptional Activity. Cancer Res Commun. 2023 Oct 6;3(10):2030-2043. [2]. WEAVER LC, et al. Toxicopathologic and pharmacologic properties of piperacetazine, a potent tranquilizing agent. Toxicol Appl Pharmacol. 1963 Jan;5:49-60. [3]. Deng J, et al. Identification of an autophagy-related gene signature for predicting prognosis and immune activity in pancreatic adenocarcinoma. Sci Rep. 2022 Apr 29;12(1):7006.
CoA	CoA of Piperacetazine

Smiles:	O=C(C1=CC=C2SC=3C=CC=CC3N(C2=C1)CCCN4CCC(CCO)CC4)C


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