PF-CBP1

PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.


Cat. No.: EX-A4474	Purity: >98%

	Chemical structure of PF-CBP1

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
500mg	825	In-stock
1g	1150	In-stock
2g	2200	In-stock
5g	4600	In-stock

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Synonyms	PF-CBP 1
CAS No.	1962928-21-7
Purity	>98%
Formula	C29H36N4O3
Mol Weight	488.6211
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Eugene L, et al. Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities. Chem Biol. 2015, 22(12):1588-1596.
CoA	CoA of PF-CBP1

Smiles:	CCCOC1=CC=C(C=C1)CCC2=NC3=C(N2CCN4CCOCC4)C=CC(=C3)C5=C(ON=C5C)C


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