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Product Information:

P2X4 antagonist-1

P2X4 antagonist-1 is a P2X4 receptor antagonist with an IC50 of 15 nM. P2X4 antagonist-1 inhibits ATP -induced calcium influx. P2X4 antagonist-1 can be used for the research of pain syndromes, endometriosis, cancer .

Cat. No.: EX-A9044    Purity: >98%
Chemical
Chemical structure of P2X4 antagonist-1


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg642In-stock
250mg1076In-stock
500mg1672In-stock
1gget quoteIn-stock


CAS No.2055601-42-6
Purity>98%
FormulaC20H15Cl3N2O4S
Mol Weight485.768
ColorWhite to off-white
Statesolid
SolubilitySoluble in DMSO
Shelf Life>3 years if stored properly
StoragePowder -20℃ 3 years, 4℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Werner S, et al. Discovery and Characterization of the Potent and Selective P2X4 Inhibitor N-[4-(3-Chlorophenoxy)-3-sulfamoylphenyl]-2-phenylacetamide (BAY-1797) and Structure-Guided Amelioration of Its CYP3A4 Induction Profile. J Med Chem. 2019 Dec 26;62(24):11194-11217.

[2]. Werner S, et al. Aromatic sulfonamide derivatives. Germany, WO2016198374 A. 2016-12-15.

CoACoA of P2X4 antagonist-1
Smiles:O=C(NC1=CC=C(OC=2C=CC=C(Cl)C2)C(=C1)S(=O)(=O)N)CC=3C(Cl)=CC=CC3Cl

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