| Synonyms | BET-IN-4 |
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| CAS No. | 1801503-93-4 |
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| Purity | >98% |
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| Formula | C22H21N3O3 |
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| Mol Weight | 375.4204 |
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| Color | Off-white to light yellow |
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| State | solid powder |
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| Solubility | DMSO : 8.33 mg/mL (22.25 mM; ultrasonic and warming and heat to 60?) |
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| Shelf Life | >2 years if stored properly |
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| Storage | Powder -20℃ 2 years; In solvent -20℃ 1 month; |
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| Shipping | Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs. |
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| Reference: | [1]. M Björkman et al. Abstract 4649: ODM-207, a novel BET-bromodomain inhibitor as a therapeutic approach for the treatment of prostate and breast cancer. Cancer Res. 76, 4649 (2016).
[2]. M Ameratunga et al. First-in-human Phase 1 open label study of the BET inhibitor ODM-207 in patients with selected solid tumours. Br J Cancer. 2020 Sep 29. |
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| CoA | CoA of ODM-207 |
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Inhibitor Specialist 
