OARV-771

OARV-771 is a VHL-based BET degrader (PROTAC) with improved cell permeability. OARV-771 shows DC50s of 6, 1, and 4 nM for Brd4, Brd2 and Brd3, respectively.


Cat. No.: EX-A7163	Purity: >98%

	Chemical structure of OARV-771

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	1285	Inquire
100mg	2500	Inquire
250mg	3500	Inquire
1g	4900	Inquire

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CAS No.	2683008-37-7
Purity	>98%
Formula	C49H59ClN8O8S2
Mol Weight	987.625
Color	White to off-white
State	solid powder
Solubility	Soluble in DMSO 100 mg/mL
Shelf Life	>2 years if stored properly
Storage	Powder -20°C, sealed storage, away from moisture; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Klein VG, et al. Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity. J Med Chem. 2021;64(24):18082-18101.
CoA	CoA of OARV-771


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