MSC2504877

MSC2504877 is a novel small molecule selective tankyrase inhibitor with IC50 of 0.7/0.8 nM against TNKS1/2, shows 771-fold selectivity for TNKS1 over PARP1 (IC50=0.54 uM).


Cat. No.: EX-A6933	Purity: >98%

	Chemical structure of MSC2504877

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	506	in_stock
250mg	1009	in_stock
500mg	1563	in_stock
1g	2511	in_stock
2g	3949	in_stock
3g	4756	in_stock

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CAS No.	1460286-21-8
Purity	>98%
Formula	C17H18N2O2
Mol Weight	282.337
Color	Off-white to light yellow
State	solid powder
Solubility	Soluble in DMSO 125 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder -20℃ 3 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Menon, Malini et al. A novel tankyrase inhibitor, MSC2504877, enhances the effects of clinical CDK4/6 inhibitors. Scientific reports vol. 9,1 201. 17 Jan. 2019, doi:10.1038/s41598-018-36447-4
CoA	CoA of MSC2504877

Smiles:	O=C1C2=CC=C(C)N2C=C(C3=CC=C(C(C)(O)C)C=C3)N1


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