Mizagliflozin

Mizagliflozin (DSP-3235 free base) is a potent, orally active and selective SGLT1 inhibitor, with a Ki of 27 nM for human SGLT1. Mizagliflozin displays 303-fold selectivity over SGLT2. Mizagliflozin is used as an antidiabetic agent that can modify postprandial blood glucose excursion.


Cat. No.: EX-A4127	Purity: >98%

	Chemical structure of Mizagliflozin

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	846	In-stock
250mg	1732	In-stock
500mg	2900	In-stock
1g	4276	In-stock

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Synonyms	DSP-3235 free base
Synonyms 2	KGA-3235 free base
CAS No.	666843-10-3
Purity	>98%
Formula	C28H44N4O8
Mol Weight	564.671
Color	off-white to light yellow
State	solid powder
Solubility	Soluble in DMSO/H2O
Shelf Life	>3 years if stored properly
Storage	Powder 4℃, protect from light, 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Inoue T, et al. Mizagliflozin, a novel selective SGLT1 inhibitor, exhibits potential in the amelioration of chronic constipation. Eur J Pharmacol. 2017 Jul 5;806:25-31. [2]. Ohno H, et al. Absorption, disposition, metabolism and excretion of [14C]mizagliflozin, a novel selective SGLT1 inhibitor, in rats. Xenobiotica. 2019 Apr;49(4):463-473.
CoA	CoA of Mizagliflozin

Smiles:	O=C(N)C(C)(C)CNCCCOC1=CC=C(CC2=C(C(C)C)NN=C2O[C@H]3[C@@H]([C@H]([C@@H]([C@@H](CO)O3)O)O)O)C(C)=C1


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