M77976

M77976 is a specific ATP-competitive inhibitor of PDK4 (pyruvate dehydrogenase kinase isoforms 4), with an IC50 of 648 μM. M77976 is potential for the research of obesity and diabetes .


Cat. No.: EX-A14940	Purity: >98%

	Chemical structure of M77976

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	492	In-stock
250mg	865	In-stock
500mg	1296	In-stock
1g	1778	In-stock

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CAS No.	394237-61-7
Purity	>98%
Formula	C17H16N2O3
Mol Weight	296.3205
Color	White to off-white
State	Solid
Solubility	Soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20℃, 3 years; 4℃, 2 years; In solvent -20℃, 1 year;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Kukimoto-Niino M, et al. Inhibitor-bound structures of human pyruvate dehydrogenase kinase 4. Acta Crystallogr D Biol Crystallogr. 2011 Sep;67(Pt 9):763-73.
CoA	CoA of M77976

Smiles:	COC1=CC=C(C=C1)C2=C(NN=C2C3=CC=C(C=C3O)O)C


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