LML-134

LML134 (compound 18b) is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg.


Cat. No.: EX-A3164	Purity: >98%

	Chemical structure of LML-134

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	1150	In-stock
500mg	1650	In-stock
1g	2300	In-stock
5g	get quote	Inquire

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CAS No.	1542135-76-1
Purity	>98%
Formula	C19H29N5O3
Mol Weight	375.4653
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Troxler T, et al. The Discovery of LML134, a Histamine H3 Receptor Inverse Agonist for the Clinical Treatment of Excessive Sleep Disorders. ChemMedChem. 2019 Jul 3;14(13):1238-1247.
CoA	CoA of LML-134

Smiles:	O=C(OC1CCN(C2=NN(C)C(C=C2)=O)CC1)N3CCN(C4CCC4)CC3


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