background


Product Information:

LDN-209929 dihydrochloride

LDN-209929 dihydrochloride is a potent and selective haspin kinase inhibitor (IC50=55 nM) with180-fold selectivity verses DYRK2 (IC50=9.9 μM). LDN-209929 is a optimized analogue of LDN-192960 .

Cat. No.: EX-A7219A    Purity: >98%
Chemical
Chemical structure of LDN-209929 dihydrochloride


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder


CAS No.1784281-97-5
Purity>98%
FormulaC17H18Cl2N2OS
Mol Weight369.309
ColorYellow to orange
Statesolid powder
SolubilityDMSO : 33.33 mg/mL
Shelf Life>2 years if stored properly
Storage4°C, sealed storage, away from moisture
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1].Gregory D Cuny, et al. Structure-activity Relationship Study of Acridine Analogs as Haspin and DYRK2 Kinase Inhibitors. Bioorg Med Chem Lett

[2].Katrin Kestav, et al. Structure, Roles and Inhibitors of a Mitotic Protein Kinase Haspin. Curr Med Chem. 2017;24(21):2276-2293.

CoACoA of LDN-209929 dihydrochloride

KEYWORDS: buy LDN-209929 dihydrochloride | LDN-209929 dihydrochloride supplier | purchase | cost | manufacturer | order | distributor | buy 1784281-97-5 | 1784281-97-5 supplier