JCN037

JCN037 (JGK037) is potent, non-covalent and brain-penetrant inhibitor of EGFR tyrosine kinase with IC50 of 2.49 nM, 3.95 nM, 4.48 nM for EGFR, p-wtEGFR and pEGFRvⅢ, respectively.


Cat. No.: EX-A5347	Purity: >98%

	Chemical structure of JCN037

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	550	In-stock
100mg	785	In-stock
200mg	1185	In-stock
500mg	1785	In-stock
1g	2585	In-stock

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CAS No.	2305154-31-6
Purity	>98%
Formula	C16H11BrFN3O2
Mol Weight	376.18
Color	Off-white to light yellow
State	solid powder
Solubility	Soluble in DMSO 50 mg/mL
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Jonathan E. Tsang, et al. Development of a Potent Brain-Penetrant EGFR Tyrosine Kinase Inhibitor against Malignant Brain Tumors. ACS Med. Chem. Lett. 2020. May 1.
CoA	CoA of JCN037


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