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Product Information:

GSK690 hydrochloride

GSK 690 (Hydrochloride) is a reversible inhibitor of lysine specific demethylase 1 (LSD1), with a Kd value of 9 nM and a biochemical IC50 of 37 nM.

Cat. No.: EX-A8792    Purity: >98%
Chemical
Chemical structure of GSK690 hydrochloride


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
50mg517in_stock
100mg827in_stock
250mg1585in_stock
500mg2570in_stock
1g4250in_stock
2g6488in_stock


SynonymsGSK-690 hydrochloride
Synonyms 2GSK690 hydrochloride
CAS No.2436760-79-9
Purity>98%
FormulaC24H24ClN3O
Mol Weight405.92
Colorlight yellow to yellow
Statesolid powder
SolubilityDMSO : 125 mg/mL
Shelf Life>2 years if stored properly
StoragePowder 4℃, sealed storage, away from moisture 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Mould DP, et al. Development of (4-Cyanophenyl)glycine Derivatives as Reversible Inhibitors of Lysine Specific Demethylase 1. J Med Chem. 2017 Oct 12;60(19):7984-7999.

[2]. Haydn T, et al. Concomitant epigenetic targeting of LSD1 and HDAC synergistically induces mitochondrial apoptosis in rhabdomyosarcoma cells. Cell Death Dis. 2017 Jun 15;8(6):e2879.

CoACoA of GSK690 hydrochloride
Smiles:N#CC1=CC=C(C2=CC(OC[C@H]3CNCC3)=CN=C2C4=CC=C(C)C=C4)C=C1.Cl

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