GSK-864

GSK864 is an isocitrate dehydrogenase 1 (IDH1) mutant inhibitor; inhibits IDH1 mutants R132C, R132H, and R132G with IC50 values of 8.8, 15.2 and 16.6 nM.


Cat. No.: EX-A4981	Purity: >98%

	Chemical structure of GSK-864

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	769	in_stock
100mg	1017	in_stock
250mg	1447	in_stock
500mg	2493	in_stock
1g	3936	in_stock
5g	13701	in_stock

Send PO to E-mail:[email protected]; or Fax:+86 020 81619670

Discount Request


Synonyms	GSK864
CAS No.	1816331-66-4
Purity	>98%
Formula	C30H31FN6O4
Mol Weight	558.6033
Color	Light brown to brown
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Okoye-Okafor UC, et al. New IDH1 mutant inhibitors for treatment of acute myeloid leukemia. Nat Chem Biol. 2015 Nov;11(11):878-86.
CoA	CoA of GSK-864

Smiles:	CC1=CC(=CC(=C1OC)C)NC(=O)C2=NN(C3=C2CN(C[C@]3(C)C(=O)N)C(=O)C4=CC=CN4)CC5=CC=C(C=C5)F


		Search