Giredestrant tartrate

Giredestrant tartrate (GDC-9545 tartrate), a non-steroidal ER ligand, is an orally active and selective estrogen receptor (ER) antagonist. Giredestrant tartrate potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Anti-tumor activity.


Cat. No.: EX-A3541A	Purity: >98%

	Chemical structure of Giredestrant tartrate

For research only, Do not use for Human!

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Synonyms	GDC-9545 tartrate
Synonyms 2	RG6171 tartrate
CAS No.	2407529-33-1
Purity	>98%
Formula	C31H37F5N4O7
Mol Weight	672.6401
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. C Metcalfe, et al. Abstract P5-04-07: GDC-9545: A novel ER antagonist and clinical candidate that combines desirable mechanistic and pre-clinical DMPK attributes.
CoA	CoA of Giredestrant tartrate

Smiles:	C[C@H](C1)N(CC(F)(F)CO)[C@H](C2=C(F)C=C(NC3CN(CCCF)C3)C=C2F)C4=C1C5=C(N4)C=CC=C5.OC([C@H](O)[C@@H](O)C(O)=O)=O


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