GCPII-IN-1 TFA

GCPII-IN-1 (Compound 2) TFA is a GCPII (also known as PSMA) inhibitor with a Ki of 44.3 nM. GCPII-IN-1 TFA can be used in the research of prostate cancer.


Cat. No.: EX-A10938	Purity: >98%

	Chemical structure of GCPII-IN-1 TFA

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
500mg	550	Inquire
1g	780	Inquire
5g	2350	Inquire

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CAS No.	1269794-89-9
Purity	>98%
Formula	C14H22F3N3O9
Mol Weight	433.3344
Color	White to off-white
State	Solid
Solubility	H2O : 160 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder 4℃, sealed storage, away from moisture and light; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Jan Tykvart, et al. Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery. Bioorg Med Chem. 2014 Aug 1;22(15):4099-108. [2]. John V. Frangioni, et al. Zwitterionic metal chelators. US20250082792A1. 2025-10-14. [3]. Mukesh K. Pandey, et al. Platform approach f-18 radiolabeling of various peptides in aqueous medium. WO2025054616A1.
CoA	CoA of GCPII-IN-1 TFA

Smiles:	OC(C(F)(F)F)=O.NCCCC[C@@H](C(O)=O)NC(N[C@H](C(O)=O)CCC(O)=O)=O


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