EPZ011989

EPZ011989 is a potent and orally active Zeste Homolog 2 (EZH2) inhibitor with metabolic stability. EPZ011989 has inhibitory inhibition for EZH2 with a Ki value of <3 nM.


Cat. No.: EX-A1583	Purity: >98%

	Chemical structure of EPZ011989

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	821	in_stock
500mg	1310	in_stock
1g	1844	in_stock
2g	3296	in_stock
5g	5253	in_stock

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CAS No.	1598383-40-4
Purity	>98%
Formula	C35H51N5O4
Mol Weight	605.8105
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Campbell JE, et al. EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity. ACS Med Chem Lett. 2015 Mar 4;6(5):491-495.
CoA	CoA of EPZ011989

Smiles:	CCN([C@H]1CC[C@@H](CC1)N(C)CCOC)C1=C(C)C(=CC(=C1)C#CCN1CCOCC1)C(=O)NCC1=C(C)C=C(C)NC1=O


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