Enerisant

Enerisant is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2.89 nM and 14.5 nM against human and rat histamine H3 receptors, respectively.


Cat. No.: EX-A10833	Purity: >98%

	Chemical structure of Enerisant

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	800	In-stock
250mg	1150	In-stock
1g	3320

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Synonyms	TS-091
CAS No.	1152747-82-4
Purity	>98%
Formula	C22H30N4O3
Mol Weight	398.4986
Color	Off-white to light yellow
State	Solid
Solubility	Soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20℃ 3 years, 4℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Hino N, et al. A novel potent and selective histamine H3 receptor antagonist enerisant: in vitro profiles, in vivo receptor occupancy, and wake-promoting and procognitive effects in rodents. Journal of Pharmacology and Experimental Therapeutics, 2020, 375(2): 276-285.
CoA	CoA of Enerisant

Smiles:	O=C(C1=CN(C2=CC=C(OCCCN3[C@H](C)CCC3)C=C2)N=C1)N4CCOCC4


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