EML4-ALK kinase inhibitor 1

EML4-ALK kinase inhibitor 1 is a potent orally active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK), with an IC50 of 1 nM.


Cat. No.: EX-A12336	Purity: >98%

	Chemical structure of EML4-ALK kinase inhibitor 1

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	480	In-stock
50mg	740	In-stock
100mg	1100	In-stock
250mg	1780	In-stock
500mg	2600	In-stock
1g	4550	In-stock

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CAS No.	1373409-08-5
Purity	>98%
Formula	C31H48N8O3
Mol Weight	580.7646
Color	Light yellow to yellow
State	Solid
Solubility	DMSO : 110 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder -20°C, sealed storage, away from moisture and light; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Iikubo K, et al. Synthesis and structure-activity relationships of pyrazine-2-carboxamide derivatives as novel echinoderm microtubule-associated protein-like 4 (EML4)-anaplastic lymphoma kinase (ALK) inhibitors. Bioorg Med Chem. 2019 Apr 15;27(8):1683-169
CoA	CoA of EML4-ALK kinase inhibitor 1

Smiles:	N(C=1C(C(N)=O)=NC(CC)=C(N[C@@H]2CC[C@@H](OC)CC2)N1)C3=CC(OC)=C(C=C3)N4CCC(CC4)N5CCN(C)CC5


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