DS17701585

DS17701585 (Compound 11) is a highly selective, orally active EP300 and CBP inhibitor with IC50 values of 0.040, 0.15, 0.45 and 0.70 µM against CBP, EP300, H3K27 and SOX2. DS17701585 can be used for cancer research.


Cat. No.: EX-A11768	Purity: >98%

	Chemical structure of DS17701585

For research only, Do not use for Human!

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CAS No.	2983027-66-1
Purity	>98%
Formula	C24H26N4O5S
Mol Weight	482.552
State	solid
Shelf Life	>3 years if stored properly
Storage	Powder 4℃, 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Kanada R, et al. Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring. Bioorg Med Chem Lett. 2022 Jun 15;66:128726.
CoA	CoA of DS17701585

Smiles:	C(=O)(C1(CCCC1)C2=CC=C(OC)C=C2)N3[C@@H](C(NC4=C5C(NN=C5)=CC=C4)=O)CS(=O)(=O)C3


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