DKFZ-251

DKFZ-251 is a potent inhibitor of kallikrein-related peptidase 6 with on-target cellular activity. DKFZ-251 demonstrated good selectivity for KLK6 compared to other KLKs, and on-target activity in a cellular assay.


Cat. No.: EX-A8454	Purity: >98%

	Chemical structure of DKFZ-251

For research only, Do not use for Human!

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CAS No.	2222059-70-1
Purity	>98%
Formula	C24H24N4O3
Mol Weight	416.4724
Color	White to off-white
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20°C, 3 years ; In solvent -20°C, 1 month
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. De Vita E, Schüler P, Lovell S, et al. Depsipeptides Featuring a Neutral P1 Are Potent Inhibitors of Kallikrein-Related Peptidase 6 with On-Target Cellular Activity. J Med Chem. 2018;61(19):8859-8874.
CoA	CoA of DKFZ-251

Smiles:	CC(NC1=C2C=CC=C1)=C2CC(OCC(NC3=C(C)N(C4=CC=CC=C4)N=C3C)=O)=O


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