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Product Information:

CDK12-IN-4

CDK12-IN-4, a pyrazolotriazine, is a potent CDK12 inhibitor with an IC50 of 0.641 μM at high ATP (2 mM). CDK12-IN-4 has no effect on CDK2/Cyclin E (IC50>20 μM) and CDK9/Cyclin T1 (IC50>20 μM) at high ATP (2 mM) (WO2021116178A1).

Cat. No.: EX-A13849    Purity: >98%
Chemical
Chemical structure of CDK12-IN-4


For research only, Do not use for Human!

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CAS No.2651196-69-7
Purity>98%
FormulaC20H20F2N8O
Mol Weight426.4226
StoragePlease store the product under the recommended conditions in the Certificate of Analysis.
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Kai Thede, et al. Pyrazolotriazines. WO2021116178A1.

CoACoA of CDK12-IN-4
Smiles:FC1=C(F)C2=C(N=C(CNC3=NC(N4CCOCC4)=NC5=C(C6CC6)C=NN35)N2)C=C1

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