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Product Information:

CBP-IN-1

CBP-IN-1 (compound 12) is a potent CBP inhibitor, with an IC50 of 1.5 nM. CBP-IN-1 also inhibits CBP BRET and BRD4(1), with IC50 values of 690 and 3100 nM, respectively.

Cat. No.: EX-A6628    Purity: >98%
Chemical
Chemical structure of CBP-IN-1


For research only, Do not use for Human!

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SynonymsCBP inhibitor (compound 12)
CAS No.1936431-44-5
Purity>98%
FormulaC27H33F2N7O
Mol Weight509.594
Statesolid powder
SolubilitySoluble in DMSO
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Romero FA, et al. GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP). J Med Chem. 2017 Nov 22;60(22):9162-9183.

CoACoA of CBP-IN-1

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