BMS-986158

BMS-986158 is a potent BET inhibitor with IC50s of 6.6 and 5 nM in NCI-H211 small cell lung cancer (SCLC) cells and MDA-MB231 triple negative breast cancer (TNBC) cells, respectively.


Cat. No.: EX-A2678	Purity: >98%

	Chemical structure of BMS-986158

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	700	In-stock
50mg	900	In-stock
100mg	1200	In-stock
250mg	1800	In-stock
1g	3300	In-stock
5g	get quote	Inquire

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CAS No.	1800340-40-2
Purity	>98%
Formula	C30H33N5O2
Mol Weight	495.6153
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Yin M, et al. Potent BRD4 inhibitor suppresses cancer cell-macrophage interaction. Nat Commun. 2020 Apr 14;11(1):1833.
CoA	CoA of BMS-986158

Smiles:	CN1N=NC(C)=C1C1=CC2=C(N=C1)C1=CC=C(C=C1N2[C@@H](C1CCOCC1)C1=CC=CC=C1)C(C)(C)O


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