BI-9321 trihydrochloride

BI-9321 is a potent, selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist with a Kd value of 166 nM. BI-9321 is inactive against NSD2-PWWP1 and NSD3-PWWP2. BI-9321 specifically disrupts histone interactions of the NSD3-PWWP1 domain with an IC50 of 1.2 μM in U2OS cells.


Cat. No.: EX-A7060	Purity: >98%

	Chemical structure of BI-9321 trihydrochloride

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	1000	In-stock
250mg	1700	In-stock
500mg	2600	In-stock
1g	3800	In-stock
5g	get quote	Inquire

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CAS No.	2387510-87-2
Purity	>98%
Formula	C22H24Cl3FN4
Mol Weight	469.81
Color	Light yellow to yellow
State	solid powder
Solubility	Soluble in DMSO 250 mg/mL H2O 25 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder 4°C, stored under nitrogen, away from moisture; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Böttcher J, et al. Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3. Nat Chem Biol. 2019 Aug;15(8):822-829.
CoA	CoA of BI-9321 trihydrochloride


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