BI-187004

BI-187004, also known as VTP-34072, is an 11β-hydroxysteroid dehydrogenase 1 inhibitor. BI187004 is being studied for the treatment of type 2 diabetes and metabolic syndrome.


Cat. No.: EX-A7115	Purity: >98%

	Chemical structure of BI-187004

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	685	Inqurie
50mg	900	Inqurie
100mg	1600	In-stock
250mg	2800	In-stock
500mg	get quote	In-stock
1g	get quote	In-stock

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Synonyms	VTP-34072
CAS No.	1303515-32-3
Purity	>98%
Formula	C21H18N4O
Mol Weight	342.3938
Color	White to off-white
State	solid powder
Solubility	Soluble in DMSO 125 mg/mL
Shelf Life	>3 years if stored properly
Storage	Powder -20℃ 3 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Maw, Hlaing H et al. N-Methylation of BI 187004 by Thiol S-Methyltransferase. Drug metabolism and disposition: the biological fate of chemicals vol. 46,6 (2018): 770-778. [2]. Bianzano, Susanna et al. Safety, tolerability, pharmacokinetics and pharmacodynamics of single oral doses of BI 187004, an inhibitor of 11beta-hydroxysteroid dehydrogenase-1, in healthy male volunteers with overweight or obesity. Clinical diabetes and endocrinology vol. 7,1 16. 15 Aug. 2021
CoA	CoA of BI-187004


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