B-HT 933 dihydrochloride

Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively[1]. Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM)[2].


Cat. No.: EX-A15280	Purity: >98%

	Chemical structure of B-HT 933 dihydrochloride

For research only, Do not use for Human!

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Synonyms	B-HT 933 dihydrochloride
Synonyms 2	Oxazoloazepin dihydrochloride
CAS No.	36067-72-8
Purity	>98%
Formula	C9H17Cl2N3O
Mol Weight	254.157
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Altamirano-Espinoza AH, et al. Specific role of α2A - and α2B -, but not α2C -, adrenoceptor subtypes in the inhibition of the vasopressor sympathetic out-flow in diabetic pithed rats. Basic Clin Pharmacol Toxicol. 2015;117(1):31-38.
CoA	CoA of B-HT 933 dihydrochloride

Smiles:	CCN1CCC2=C(CC1)OC(=N2)N.Cl.Cl


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