ARD-266

ARD-266 is a highly potent and von Hippel-Lindau E3 ligase-based Androgen Receptor (AR) PROTAC degrader. ARD-266 effectively induces degradation of AR protein in AR-positive LNCaP, VCaP, and 22Rv1 prostate cancer cell lines with DC50 values of 0.2-1 nM.


Cat. No.: EX-A5712	Purity: >98%

	Chemical structure of ARD-266

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	782	In-stock
100mg	get quote	In-stock
250mg	get quote	In-stock
500mg	get quote	In-stock
1g	get quote	In-stock
2g	get quote	In-stock

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CAS No.	2666951-70-6
Purity	>98%
Formula	C52H59ClN6O7
Mol Weight	915.514
Color	White to off-white
State	solid powder
Solubility	Soluble in DMSO 100 mg/mL
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Han X, et al. Discovery of Highly Potent and Efficient PROTAC Degraders of Androgen Receptor (AR) by Employing Weak Binding Affinity VHL E3 Ligase Ligands. J Med Chem. 2019 Dec 26;62(24):11218-11231.
CoA	CoA of ARD-266


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