AG-041R

AG-041R is a potent and selective CCK2 Receptor/Gastrin antagonist. AG-041R inhibits gastrin-evoked secretion of pancreastatin with an IC50 of 2.2 nM. AG-041R inhibits cell growth of Mastomys ECL carcinoid tumor cells .


Cat. No.: EX-A15143	Purity: >98%

	Chemical structure of AG-041R

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	1580	Inquire
100mg	1900	Inquire
250mg	get quote	Inquire
500mg	get quote	Inquire
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CAS No.	159883-95-1
Purity	>98%
Formula	C31H36N4O5
Mol Weight	544.6413
Color	White to off-white
State	Solid
Shelf Life	>3 years if stored properly
Storage	Powder -20℃, 3 years; In solvent -20℃, 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Ding XQ, et al. Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: a study of their effects on rat stomach enterochromaffin-like cell activity. Pharmacol Toxicol. 1997 Nov;81(5):232-7. [2]. Lindström, E., et al. Pharmacological analysis of CCK2 receptor antagonists using isolated rat stomach ECL cells. Br. J. Pharmacol. 127(2), 530-536 (1999).
CoA	CoA of AG-041R

Smiles:	CC(C=C1)=CC=C1NC(C[C@]2(C3=CC=CC=C3N(C2=O)CC(OCC)OCC)NC(NC4=CC=C(C=C4)C)=O)=O


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