A-366

Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50 = 3.3 nM). Exhibits >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. Decreases levels of lysine 9 dimethylation on histone H3 (H3K9Me2) in PC3 cells.


Cat. No.: EX-A2328	Purity: >98%

	Chemical structure of A-366

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	785	In-stock
500mg	985	In-stock
1g	1485	In-stock
5g	get quote	In-stock
10g	get quote	Inquire

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CAS No.	1527503-11-2
Purity	>98%
Formula	C19H27N3O2
Mol Weight	329.4366
State	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Pappano WN, et al. PLoS One. 2015, 10(7):e0131716. [2]. Sweis RF, et al. ACS Med Chem Lett. 2014, 5(2):205-209.
CoA	CoA of A-366

Smiles:	COC1=CC2=C(C=C1OCCCN1CCCC1)N=C(N)C21CCC1


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