I-BET567

I-BET567 is a potent and orally active inhibitor of pan-BET candidate with pIC50s of 6.9 and 7.2 for BRD4 BD1 and BD2, respectively. I-BET567 has been demonstrated efficacy in mouse models of oncology and inflammation.


Cat. No.: EX-A10255	Purity: >98%

	Chemical structure of I-BET567

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	1150	In-stock
250mg	1900	In-stock
500mg	2785	In-stock
1g	3985	In-stock

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CAS No.	1887237-54-8
Purity	>98%
Formula	C17H18ClN5O2
Mol Weight	359.81
Appearance	white to off-white solid
Solubility	soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder 4℃,protect from light, 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Humphreys PG, et al. Design, Synthesis, and Characterization of I-BET567, a Pan-Bromodomain and Extra Terminal (BET) Bromodomain Oral Candidate [published online ahead of print, 2022 Jan 7].
CoA	CoA of I-BET567

Smiles:	O=C(C1=CC2=C(N(C(C)=O)[C@@H](C)C[C@H]2NC3=NC=C(Cl)C=N3)C=C1)N


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