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Product Information:

Encequidar mesylate

Encequidar mesylate (HM30181 mesylate) is a potent P-glycoprotein inhibitor.

Cat. No.: EX-A3429    Purity: >98%
Chemical
Chemical structure of Encequidar mesylate


For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg400In-stock
250mg685In-stock
500mg885In-stock
1g1385In-stock
2g2285In-stock
5g3885Inquire


SynonymsHM30181 mesylate
Synonyms 2HM30181A mesylate
CAS No.849675-87-2
Purity>98%
FormulaC39H40N6O10S
Mol Weight784.834
Appearancesolid powder
SolubilitySoluble in DMSO, not in water
Shelf Life>4 years if stored properly
StoragePowder 4℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Kim JC, et al. Effect of HM30181 mesylate salt-loaded microcapsules on the oral absorption of NSC 125973 as a novel P-glycoprotein inhibitor. Int J Pharm. 2016 Jun 15;506(1-2):93-101.

[2]. Joo KM, et al. Response of brain specific microenvironment to P-glycoprotein inhibitor: an important factor determining therapeutic effect of P-glycoprotein inhibitor on brain metastatic tumors. Int J Oncol. 2008 Oct;33(4):705-12.

CoACoA of Encequidar mesylate
Smiles:O=C(C1=CC(C2=CC=CC=C2O1)=O)NC3=CC(OC)=C(OC)C=C3C4=NN(C5=CC=C(CCN6CC7=C(C=C(OC)C(OC)=C7)CC6)C=C5)N=N4.CS(=O)(O)=O

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