Dersimelagon

Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively.


Cat. No.: EX-A8422	Purity: >98%

	Chemical structure of Dersimelagon

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	450	In-stock
50mg	600	In-stock
100mg	950	In-stock
200mg	1550	In-stock
500mg	get quote	In-stock
1g	get quote	In-stock

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Synonyms	MT-7117
CAS No.	1835256-48-8
Purity	>98%
Formula	C36H45F4N3O5
Mol Weight	675.7532
Appearance	Off-white to light yellow solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. T. Suzuki, et al. Melanogenic effect of dersimelagon (MT-7117), a novel oral melanocortin 1 receptor agonist. Skin Health Dis. 2022; 2(1):e78. [2]. Erwin AL, et al. Porphyrias in the Age of Targeted Therapies. Diagnostics (Basel). 2021;11(10):1795. Published 2021 Sep 29.
CoA	CoA of Dersimelagon

Smiles:	COC[C@H]1CN(C[C@@H]1C2=C(C=C(C=C2)C(F)(F)F)N3CCC(CC3)C(=O)O)C(=O)[C@@]4(CN(C[C@H]4C5=CC=C(C=C5)OC)C6CCCC6)F


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